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51-05-8, Procaine hydrochloride

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ọja Tags

Lilo Procaine hydrochloride
Procaine Hydrochloride jẹ oogun anesitetiki agbegbe ti ẹgbẹ amino ester.Target: OthersProcaine jẹ anesitetiki agbegbe ti iru ester ti o ni ibẹrẹ ti o lọra ati akoko kukuru ti igbese.Procaine (0.01-100 microM) ṣe idiwọ olugba 5-HT3- alarina lọwọlọwọ inu ni gbogbo-cell patch dimole gbigbasilẹ.Procaine han lati gbejade idinamọ idije lori awọn olugba 5-HT3 pẹlu KD ti 1.7 microM [1].Procaine jẹ oluranlowo DNA-demethylating ti o ṣe agbejade idinku 40% ninu akoonu DNA 5-methylcytosine gẹgẹbi a ti pinnu nipasẹ elekitirophoresis capillary-giga tabi tito nkan lẹsẹsẹ DNA henensiamu lapapọ.Procaine tun le demethylate densely hypermethylated CpG erekusu.Procaine tun ni awọn ipa idalọwọduro idagbasoke ninu awọn sẹẹli alakan wọnyi, ti o nfa imuni mitotic [2].Procaine n ṣiṣẹ bi itara ti awọn sẹẹli eto limbic, ati pe procaine n ṣe iyipada gbigbe synapti ni diẹ ninu awọn, ṣugbọn kii ṣe gbogbo rẹ, awọn ipa ọna ti o jade lati amygdale [3]

Awọn orukọ

Oruko Procaine hydrochloride
Itumọ Diẹ Synonyms

 Procaine hydrochloride Iṣẹ iṣe

Apejuwe Procaine Hydrochloride jẹ oogun anesitetiki agbegbe ti ẹgbẹ amino ester.Target: OthersProcaine jẹ anesitetiki agbegbe ti iru ester ti o ni ibẹrẹ ti o lọra ati akoko kukuru ti igbese.Procaine (0.01-100 microM) ṣe idiwọ olugba 5-HT3- alarina lọwọlọwọ inu ni gbogbo-cell patch dimole gbigbasilẹ.Procaine han lati gbejade idinamọ idije lori awọn olugba 5-HT3 pẹlu KD ti 1.7 microM [1].Procaine jẹ oluranlowo DNA-demethylating ti o ṣe agbejade idinku 40% ninu akoonu DNA 5-methylcytosine gẹgẹbi a ti pinnu nipasẹ elekitirophoresis capillary ti o ga julọ tabi tito nkan lẹsẹsẹ DNA lapapọ.Procaine tun le demethylate densely hypermethylated CpG erekusu.Procaine tun ni awọn ipa idalọwọduro idagbasoke ninu awọn sẹẹli alakan wọnyi, ti o nfa imuni mitotic [2].Awọn iṣẹ Procaine gẹgẹbi itara ti awọn sẹẹli eto limbic, ati pe procaine n ṣe iyipada gbigbe synapti ni diẹ ninu awọn, ṣugbọn kii ṣe gbogbo, awọn ipa ọna ti o jade lati amygdale [3].
Jẹmọ Catalog
Awọn itọkasi

[1]. Fan, P. ati FF Weight, Procaine ṣe ailagbara iṣẹ ti eka ikanni receptor-ion eka 5-HT3 ninu awọn neurons sensọ ganglion eku.Neuropharmacology, 1994. 33 (12): p.Ọdun 1573-9.

[2]. Villar-Garea, A., et al., Procaine jẹ oluranlowo DNA-demethylating pẹlu awọn ipa idilọwọ idagbasoke ninu awọn sẹẹli alakan eniyan.Akàn Res, 2003. 63 (16): p.4984-9.

[3]. Adamec, RE ati C. Stark-Adamec, Awọn ipa ti procaine HCl lori cellular olugbe ati evoked esi aṣayan iṣẹ-ṣiṣe laarin awọn limbic eto ti o nran.Ẹri fun igbese excitatory iyatọ ti procaine ni ọpọlọpọ awọn iyika limbic.Prog Neuropsychopharmacol Biol Psychiatry, 1987. 11 (4): p.345-64.

 Kemikali & Ti ara Properties

Ojuami farabale 195-196 ° C 17mm
Ojuami Iyo 155-156°C(tan.)
Ilana molikula C13H21ClN2O2
Òṣuwọn Molikula 272.771
Oju filaṣi 195-196 ° C / 17mm
Gangan Ibi 272.129150
PSA 55.56000
LogP 3.15060
Iduroṣinṣin Idurosinsin.Ibamu pẹlu awọn aṣoju oxidizing lagbara.
Omi Solubility tiotuka

 Toxicological Alaye

Ìdámọ̀ kẹ́míkà

NỌMBA RTECS:
DG2275000
ORUKO Kemikali:
Benzoic acid, p-amino-, 2- (diethylamino) ethyl ester, monohydrochloride.
NỌMBA Iforukọsilẹ CAS:
51-05-8
Imudojuiwọn Kẹhin:
Ọdun 199701
DATA NKAN TO TOKA:
27
FORMULA MOLEKU:
C13-H20-N2-O2.Cl-H
ÒṢÙN MOLEKULU:
272.81
AKIYESI ILA WISWESSER:
ZR DVO2N2 & 2 & GH

DATA EWU ILERA

TOXICITY DATA

ORISI idanwo:
TDLo – Iwọn majele ti a tẹjade ti o kere julọ
ONA TI IFIHAN:
Awọn ipa-ọna pupọ
Awọn ẹya ti a ṣe akiyesi:
Eniyan - eniyan
DOSE/AGBA:
2286 mg/kg/8D-mo
AWON IFA OLORO:
Àrùn, ureter, àpòòtọ - awọn iyipada ninu tubules (pẹlu ikuna kidirin nla, negirosisi tubular nla)
Itọkasi:
AJKDDP American Journal of Kidney Arun.(Grune & Stratton, Inc., Iwe-alabapin Iwe akosile Dept., POB 6280, Duluth, MN 55806) V.1- 1981- Iwọn didun (ọrọ) / oju-iwe / ọdun: 7,502,1986
ORISI idanwo:
LD50 – Apaniyan iwọn lilo, 50 ogorun pa
ONA TI IFIHAN:
Ẹnu
Awọn ẹya ti a ṣe akiyesi:
Rodent - eku
DOSE/AGBA:
200 mg / kg
AWON IFA OLORO:
Awọn alaye ti awọn ipa majele ko royin miiran ju iye iwọn lilo apaniyan
Itọkasi:
ZENBAX Zeitschrift fuer Naturforschung, Teil B: Anorganische Chemie, Organische Chemie, Biochemie, Biophysik, Biologie.(Tuebingen, Fed. aṣoju Ger.) V.2B-27B, 1947-1972.Fun alaye akede, wo ZNCBDA.Iwọn didun (oro)/oju-iwe/odun: 6B,183,1951
ORISI idanwo:
LD50 – Apaniyan iwọn lilo, 50 ogorun pa
ONA TI IFIHAN:
Intraperitoneal
Awọn ẹya ti a ṣe akiyesi:
Rodent - eku
DOSE/AGBA:
160 mg / kg
AWON IFA OLORO:
Awọn alaye ti awọn ipa majele ko royin miiran ju iye iwọn lilo apaniyan
Itọkasi:
KSRNAM Kiso to Rinsho.isẹgun Iroyin.(Yubunsha Co., Ltd., 1-5, Kanda Suda-Cho, Chiyoda-ku, KS Bldg., Tokyo 101, Japan) V.1- 1960- Iwọn didun (oro)/oju-iwe/odun: 13,791,1979
ORISI idanwo:
LD50 – Apaniyan iwọn lilo, 50 ogorun pa
ONA TI IFIHAN:
Subcutaneous
Awọn ẹya ti a ṣe akiyesi:
Rodent - eku
DOSE/AGBA:
597 mg / kg
AWON IFA OLORO:
Awọn alaye ti awọn ipa majele ko royin miiran ju iye iwọn lilo apaniyan
Itọkasi:
PHACAI Pharmaceutical Archives.(School of Pharmacy, University of Wisconsin, Madison, WI) V.1-16, 1898-1945.Ti dawọ duro.Iwọn didun (oro) / oju-iwe / ọdun: 11,81,1940
ORISI idanwo:
LD50 – Apaniyan iwọn lilo, 50 ogorun pa
ONA TI IFIHAN:
Iwo inu
Awọn ẹya ti a ṣe akiyesi:
Rodent - eku
DOSE/AGBA:
38 mg / kg
AWON IFA OLORO:
Ihuwasi - awọn gbigbọn tabi ipa lori ẹnu-ọna ijagba Iwa - ihamọ iṣan tabi spasticity Lungs, Thorax, tabi Respiration - awọn iyipada miiran
Itọkasi:
ANESAV Anesthesiology.(Lippincott/Harper, Journal Fulfillment Dept., 2350 Virginia Ave., Hagerstown, MD 21740) V.1- 1940- Iwọn didun (oro)/oju-iwe/odun: 3,398,1942
ORISI idanwo:
LD50 – Apaniyan iwọn lilo, 50 ogorun pa
ONA TI IFIHAN:
Ti ko royin
Awọn ẹya ti a ṣe akiyesi:
Rodent - eku
DOSE/AGBA:
150 mg / kg
AWON IFA OLORO:
Awọn alaye ti awọn ipa majele ko royin miiran ju iye iwọn lilo apaniyan
Itọkasi:
ARZNAD Arzneimittel-Forschung.Iwadi Oògùn.(Editio Cantor Verlag, Postfach 1255, W-7960 Aulendorf, Fed. Aṣoju Ger.) V.1- 1951- Iwọn didun (oro) / oju-iwe / ọdun: 17,1012,1967
ORISI idanwo:
LD50 – Apaniyan iwọn lilo, 50 ogorun pa
ONA TI IFIHAN:
Ẹnu
Awọn ẹya ti a ṣe akiyesi:
Rodent - Asin
DOSE/AGBA:
175 mg / kg
AWON IFA OLORO:
Awọn alaye ti awọn ipa majele ko royin miiran ju iye iwọn lilo apaniyan
Itọkasi:
ZENBAX Zeitschrift fuer Naturforschung, Teil B: Anorganische Chemie, Organische Chemie, Biochemie, Biophysik, Biologie.(Tuebingen, Fed. aṣoju Ger.) V.2B-27B, 1947-1972.Fun alaye akede, wo ZNCBDA.Iwọn didun (oro)/oju-iwe/odun: 6B,183,1951
ORISI idanwo:
LD50 – Apaniyan iwọn lilo, 50 ogorun pa
ONA TI IFIHAN:
Intraperitoneal
Awọn ẹya ti a ṣe akiyesi:
Rodent - Asin
DOSE/AGBA:
165 mg / kg
AWON IFA OLORO:
Awọn alaye ti awọn ipa majele ko royin miiran ju iye iwọn lilo apaniyan
Itọkasi:
ARZNAD Arzneimittel-Forschung.Iwadi Oògùn.(Editio Cantor Verlag, Postfach 1255, W-7960 Aulendorf, Fed. Aṣoju Ger.) V.1- 1951- Iwọn didun (oro) / oju-iwe / ọdun: 26,793,1976
ORISI idanwo:
LD50 – Apaniyan iwọn lilo, 50 ogorun pa
ONA TI IFIHAN:
Subcutaneous
Awọn ẹya ti a ṣe akiyesi:
Rodent - Asin
DOSE/AGBA:
339 mg / kg
AWON IFA OLORO:
Awọn alaye ti awọn ipa majele ko royin miiran ju iye iwọn lilo apaniyan
Itọkasi:
BCFAAI Bollettino Chimico Farmaceutico.(Societa Editoriale Farmaceutica, Nipasẹ Ausono 12, 20123 Milan, Italy) V.33- 1894- Iwọn didun (oro)/oju-iwe/odun: 107,310,1968
ORISI idanwo:
LD50 – Apaniyan iwọn lilo, 50 ogorun pa
ONA TI IFIHAN:
Iwo inu
Awọn ẹya ti a ṣe akiyesi:
Rodent - Asin
DOSE/AGBA:
33 mg / kg
AWON IFA OLORO:
Awọn alaye ti awọn ipa majele ko royin miiran ju iye iwọn lilo apaniyan
Itọkasi:
ANPRBG Ilọsiwaju anesthesia.(Elsevier Science Publishing Co., Inc., 655 Avenue of the Americas, New York, NY 10010) V.13- 1966- Iwọn didun (oro)/oju-iwe/odun: 36,79,1989
ORISI idanwo:
LD50 – Apaniyan iwọn lilo, 50 ogorun pa
ONA TI IFIHAN:
inu iṣan
Awọn ẹya ti a ṣe akiyesi:
Rodent - Asin
DOSE/AGBA:
500 mg / kg
AWON IFA OLORO:
Awọn alaye ti awọn ipa majele ko royin miiran ju iye iwọn lilo apaniyan
Itọkasi:
THERAP Itọju ailera.(Doin, Editeurs, 8, Place de l'Odeon, F-75006 Paris, France) V.1- 1946- Iwọn didun (ọrọ)/oju-iwe/ọdun: 9,332,1954
ORISI idanwo:
LD50 – Apaniyan iwọn lilo, 50 ogorun pa
ONA TI IFIHAN:
Intracerebral
Awọn ẹya ti a ṣe akiyesi:
Rodent - Asin
DOSE/AGBA:
33 mg / kg
AWON IFA OLORO:
Awọn alaye ti awọn ipa majele ko royin miiran ju iye iwọn lilo apaniyan
Itọkasi:
NYKZAU Nippon Yakurigaku Zasshi.Iwe akọọlẹ Japanese ti Pharmacology.(Nippon Yakuri Gakkai, c/o Kyoto Daigaku Igakubu Yakurigaku Kyoshitsu, Konoe-cho, Yoshida, Sakyo-ku, Kyoto 606, Japan) V.40- 1944- Iwọn didun (ọrọ)/oju-iwe/odun: 63(3),93S Ọdun 1967
ORISI idanwo:
LD50 – Apaniyan iwọn lilo, 50 ogorun pa
ONA TI IFIHAN:
Òbí
Awọn ẹya ti a ṣe akiyesi:
Rodent - Asin
DOSE/AGBA:
192 mg / kg
AWON IFA OLORO:
Ihuwasi – ijagba tabi ipa lori iloro ijagba Iwa – itara ẹdọforo, Thorax, tabi Respiration – dyspnea
Itọkasi:
Awọn egboogi ANTCAO ati Chemotherapy (Washington, DC).(Washington, DC) V.1-12, 1951-62.Fun alaye akede, wo CLMEA3.Iwọn didun (ọrọ) / oju-iwe / ọdun: 4,633,1954
ORISI idanwo:
LD50 – Apaniyan iwọn lilo, 50 ogorun pa
ONA TI IFIHAN:
Iwo inu
Awọn ẹya ti a ṣe akiyesi:
Mammal – aja
DOSE/AGBA:
63 mg / kg
AWON IFA OLORO:
Arun ọkan - awọn iyipada miiran Vascular – BP sokale ko ṣe afihan ni apakan autonomic Awọn ẹdọforo, Thorax, tabi Respiration - ibanujẹ atẹgun
Itọkasi:
JDREAF Journal of Dental Research.(International Assoc. fun Dental Research, 734 15th St., NW, Suite 809, Washington, DC 20005) V.1- 1919- Iwọn didun (oro)/oju-iwe/odun: 20,425,1941
ORISI idanwo:
LDLo – Iwọn apaniyan ti a tẹjade ti o kere julọ
ONA TI IFIHAN:
Intracerebral
Awọn ẹya ti a ṣe akiyesi:
Mammal – aja
DOSE/AGBA:
11 mg / kg
AWON IFA OLORO:
Awọn alaye ti awọn ipa majele ko royin miiran ju iye iwọn lilo apaniyan
Itọkasi:
ARZNAD Arzneimittel-Forschung.Iwadi Oògùn.(Editio Cantor Verlag, Postfach 1255, W-7960 Aulendorf, Fed. Aṣoju Ger.) V.1- 1951- Iwọn didun (oro) / oju-iwe / ọdun: 9,137,1959
ORISI idanwo:
LDLo – Iwọn apaniyan ti a tẹjade ti o kere julọ
ONA TI IFIHAN:
Iwo inu
Awọn ẹya ti a ṣe akiyesi:
Mammal – ologbo
DOSE/AGBA:
10 mg / kg
AWON IFA OLORO:
Iwa - gbigbọn tabi ipa lori ẹnu-ọna ijagba Cardiac - iyipada ni oṣuwọn
Itọkasi:
Iwe akọọlẹ JPETAB ti Ẹkọ nipa oogun ati Awọn Iwosan Imọran.(Williams & Wilkins Co., 428 E. Preston St., Baltimore, MD 21202) V.1- 1909/10- Iwọn didun (oro)/oju-iwe/odun: 8,385,1916
ORISI idanwo:
LD50 – Apaniyan iwọn lilo, 50 ogorun pa
ONA TI IFIHAN:
Subcutaneous
Awọn ẹya ti a ṣe akiyesi:
Rodent - ehoro
DOSE/AGBA:
687 mg / kg
AWON IFA OLORO:
Awọn alaye ti awọn ipa majele ko royin miiran ju iye iwọn lilo apaniyan
Itọkasi:
Iwe akọọlẹ JPETAB ti Ẹkọ nipa oogun ati Awọn Iwosan Imọran.(Williams & Wilkins Co., 428 E. Preston St., Baltimore, MD 21202) V.1- 1909/10- Iwọn didun (oro)/oju-iwe/odun: 93,388,1948
ORISI idanwo:
LD50 – Apaniyan iwọn lilo, 50 ogorun pa
ONA TI IFIHAN:
Iwo inu
Awọn ẹya ti a ṣe akiyesi:
Rodent - ehoro
DOSE/AGBA:
43 mg / kg
AWON IFA OLORO:
Awọn alaye ti awọn ipa majele ko royin miiran ju iye iwọn lilo apaniyan
Itọkasi:
KSRNAM Kiso to Rinsho.isẹgun Iroyin.(Yubunsha Co., Ltd., 1-5, Kanda Suda-Cho, Chiyoda-ku, KS Bldg., Tokyo 101, Japan) V.1- 1960- Iwọn didun (oro)/oju-iwe/odun: 13,791,1979
ORISI idanwo:
LD50 – Apaniyan iwọn lilo, 50 ogorun pa
ONA TI IFIHAN:
Intracerebral
Awọn ẹya ti a ṣe akiyesi:
Rodent - ehoro
DOSE/AGBA:
4800 iwon / kg
AWON IFA OLORO:
Ihuwasi - gbigbọn tabi ipa lori iloro ijagba Iwa - ataxia Lungs, Thorax, tabi Respiration - dyspnea
Itọkasi:
ARZNAD Arzneimittel-Forschung.Iwadi Oògùn.(Editio Cantor Verlag, Postfach 1255, W-7960 Aulendorf, Fed. Aṣoju Ger.) V.1- 1951- Iwọn didun (oro) / oju-iwe / ọdun: 9,137,1959
ORISI idanwo:
LD50 – Apaniyan iwọn lilo, 50 ogorun pa
ONA TI IFIHAN:
Ti ko royin
Awọn ẹya ti a ṣe akiyesi:
Rodent - ehoro
DOSE/AGBA:
41 mg / kg
AWON IFA OLORO:
Awọn alaye ti awọn ipa majele ko royin miiran ju iye iwọn lilo apaniyan
Itọkasi:
ARZNAD Arzneimittel-Forschung.Iwadi Oògùn.(Editio Cantor Verlag, Postfach 1255, W-7960 Aulendorf, Fed. Aṣoju Ger.) V.1- 1951- Iwọn didun (oro)/oju-iwe/odun: 24,1957,1974
ORISI idanwo:
LDLo – Iwọn apaniyan ti a tẹjade ti o kere julọ
ONA TI IFIHAN:
Intraspinal
Awọn ẹya ti a ṣe akiyesi:
Rodent - ehoro
DOSE/AGBA:
15504 iwon / kg
AWON IFA OLORO:
Nafu Agbeegbe ati Aibalẹ – Anesitetiki agbegbe
Itọkasi:
ANESAV Anesthesiology.(Lippincott/Harper, Journal Fulfillment Dept., 2350 Virginia Ave., Hagerstown, MD 21740) V.1- 1940- Iwọn didun (oro)/oju-iwe/odun: 1,305,1940
ORISI idanwo:
LD50 – Apaniyan iwọn lilo, 50 ogorun pa
ONA TI IFIHAN:
Subcutaneous
Awọn ẹya ti a ṣe akiyesi:
Rodent - Guinea ẹlẹdẹ
DOSE/AGBA:
407 mg / kg
AWON IFA OLORO:
Awọn alaye ti awọn ipa majele ko royin miiran ju iye iwọn lilo apaniyan
Itọkasi:
Iwe akọọlẹ JPETAB ti Ẹkọ nipa oogun ati Awọn Iwosan Imọran.(Williams & Wilkins Co., 428 E. Preston St., Baltimore, MD 21202) V.1- 1909/10- Iwọn didun (oro)/oju-iwe/odun: 93,388,1948
ORISI idanwo:
LD50 – Apaniyan iwọn lilo, 50 ogorun pa
ONA TI IFIHAN:
Iwo inu
Awọn ẹya ti a ṣe akiyesi:
Rodent - Guinea ẹlẹdẹ
DOSE/AGBA:
51 mg / kg
AWON IFA OLORO:
Awọn alaye ti awọn ipa majele ko royin miiran ju iye iwọn lilo apaniyan
Itọkasi:
AIPTAK Archives Internationales de Pharmacodynamie et de Therapie.(Heymans Institute of Pharmacology, De Pintelaan 185, B-9000 Ghent, Belgium) V.4- 1898- Iwọn didun (oro) / oju-iwe / ọdun: 113,313,1958 DATA IWỌRỌ : NOHS – Iwadii Ewu ti Iṣẹ iṣe ti Orilẹ-ede (1974) NOHS koodu Ewu – 83464 Nọmba ti Awọn ohun elo: 93 (iṣiro) Nọmba ti Awọn ile-iṣẹ: 2 No. Iwadi Iṣafihan Iṣẹ iṣe (1983) NOES koodu ewu - 83464 No. ti Awọn ohun elo: 489 (iṣiro) Bẹẹkọ ti Awọn ile-iṣẹ: 3 Nọmba ti Awọn iṣẹ: 13 No. )

 Alaye Aabo

Aami GHS06
GHS06
Ọrọ ifihan agbara Ijamba
Ewu Gbólóhùn H301-H317
Awọn Gbólóhùn Iṣọra P280-P301 + P310
Ohun elo Idaabobo Ti ara ẹni Awọn iboju oju; Awọn iboju oju; Awọn ibọwọ; iru P2 (EN 143) awọn katiriji atẹgun
Awọn koodu ewu T: Majele
Awọn gbolohun ọrọ ewu R25; R36/37/38
Awọn gbolohun Aabo S36 / 37/39-S45-S37 / 39-S26
RIDADR UN 2811 6.1/PG 3
WGK Germany 3
RTECS DG2275000
Ẹgbẹ apoti III
Kíláàsì ewu 6.1
HS koodu 2922499100

 Precursor & DownStream

Precursor 0
DownStream 2

 Awọn kọsitọmu

HS koodu 2922499990
Lakotan HS:2922499990 awọn amino acids miiran, yatọ si awọn ti o ni diẹ ẹ sii ju iru iṣẹ atẹgun, ati awọn esters wọn;iyọ ti VAT:17.0% Oṣuwọn idinku owo-ori:9.0% Awọn ipo abojuto:AB(iwe-ẹri ti ayewo fun awọn ọja inu, iwe-ẹri ti ayewo fun awọn ọja ita) Owo idiyele MFN: 6.5% Owo-ori gbogbogbo: 30.0%

 Ìwé40

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Awọn aaye pipo ti elekitirolisisi ni awọn iyọkuro elekitiromembrane ti ekikan ati awọn itupalẹ ipilẹ.

Anali.Chim.Ìṣirò 887, 92-100, (2015)

Electrolysis wa ni ibi gbogbo ni gbogbo awọn ilana elekitirokemika pẹlu isediwon elekitiromembrane (EME).Awọn ipa ti electrolysis lori awọn aaye pipo ti EME ni a ṣe ayẹwo ni kikun fun…

 Awọn itumọ ọrọ sisọ

dajudaju
Procaine (hydrochloride)
Procaine hydrochloride
Jenacaine
novocaine hydrochloride
Procaine, hydrochloride
procaine HCl
ethocaine
2- (Diethylamino) ethyl-4-aminobenzolcarboxylathydrochlorid
eugerase
Isocaine-Asid
Benzoic acid, 4-amino-, 2- (diethylamino) ethyl ester, hydrochloride (1:1)
MFCD00007893
2- (Diethylamino) ethyl-4-aminobenzoathydrochlorid
2- (Diethylamino) ethyl 4-aminobenzoate hydrochloride (1: 1)
4-Aminobenzoic Acid 2- (Diethylamino) ethyl Ester Hydrochloride
naucaine
Alocaine
2- (diethylamino) ethyl 4-aminobenzoate hydrochloride
EINECS 200-077-2
Bernacaine
anestil
anadolor
p-aminobenzoyldiethylaminoethanol hydrochloride
paracain
irokaini
2-Diethylaminoethyl 4-aminobenzoate hydrochloride
syncaine
4-Aminobenzoate de 2-(diéthylamino)éthyle chlorhydrate
topukain

 

 

 

Lilo Procaine hydrochloride
Procaine Hydrochloride jẹ oogun anesitetiki agbegbe ti ẹgbẹ amino ester.Target: OthersProcaine jẹ anesitetiki agbegbe ti iru ester ti o ni ibẹrẹ ti o lọra ati akoko kukuru ti igbese.Procaine (0.01-100 microM) ṣe idiwọ olugba 5-HT3- alarina lọwọlọwọ inu ni gbogbo-cell patch dimole gbigbasilẹ.Procaine han lati gbejade idinamọ idije lori awọn olugba 5-HT3 pẹlu KD ti 1.7 microM [1].Procaine jẹ oluranlowo DNA-demethylating ti o ṣe agbejade idinku 40% ninu akoonu DNA 5-methylcytosine gẹgẹbi a ti pinnu nipasẹ elekitirophoresis capillary-giga tabi tito nkan lẹsẹsẹ DNA henensiamu lapapọ.Procaine tun le demethylate densely hypermethylated CpG erekusu.Procaine tun ni awọn ipa idalọwọduro idagbasoke ninu awọn sẹẹli alakan wọnyi, ti o nfa imuni mitotic [2].Procaine n ṣiṣẹ bi itara ti awọn sẹẹli eto limbic, ati pe procaine n ṣe iyipada gbigbe synapti ni diẹ ninu awọn, ṣugbọn kii ṣe gbogbo rẹ, awọn ipa ọna ti o jade lati amygdale [3]


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